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. Author manuscript; available in PMC: 2022 Jan 19.
Published in final edited form as: ChemMedChem. 2020 Oct 23;16(2):335–339. doi: 10.1002/cmdc.202000726

Table 1.

Antiribosomal Activities and Selectivities.

IC50 [μM] Selectivity
Strain wt Mit13 A1555G Cyt14 Mit13 A1555G Cyt14
Apramycin 0.15±0.05 119±30 98±33 129±26 793 653 860
2 0.071±0.015 68±20 13±3 190±105 957 183 2676
3 0.052±0.026 118±34 99±22 97±14 2269 1904 1865
4 0.032±0.014 43±7 21±3 40±7 1343 656 1250