Table 2.
The inhibitors partially or completely acting on TRAP1.
Drug | Structure | Properties | Types of cancer | Refs. |
---|---|---|---|---|
Gamitrinib-G4 |
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Hsp90 inhibitor and TRAP1 inhibitor | Prostate cancer | (74) |
Shepherdin |
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Hsp90 inhibitor and TRAP1 inhibitor | Glioblastoma, retinoblastoma | (75, 76) |
DN401 |
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Strong TRAP1 inhibitor but weak Hsp90 inhibitor | Cervical cancer, liver cancer, brain cancer, kidney cancer, lung cancer, prostate cancer | (77, 78) |
Honokiol bis-dichloroacetate (HDCA) |
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TRAP1-specific inhibitor | (79) |