TABLE 2.

Agonists at A_2A-adenosine receptors.

Agonist name	Ki nM
Adenosine	310		Fredholm et al. (2011)
CGS 21680	27		Fredholm et al. (2011)
	1,570 canine		Glover et al., 2001
UK-432097	4		Fredholm et al. (2011)
ATL-146e (Apadenoson)	0.5		Fredholm et al. (2011)
	44 canine		Glover et al. (2001)
MRE 0094 (sonedenoson)	ND		Fredholm et al. (2011)
(CV-3146) regadenoson	290		Fredholm et al. (2011)
BVT 115959	Not disclosed		https://clinicaltrials.gov/search/intervention = BVT.115959
NECA	9.7		Fredholm et al. (2011)
HE-NECA	2.2		Darbousset et al. (2014)
(WRC-0470) binodenoson	290		Fredholm et al. (2011)
WRC-0090			Shryock and Belardinelli (1997)
WRC-0013			Shryock and Belardinelli (1997)
UK371104	Anti lg 7.7		Jacobson et al. (2019)
GW328267X	Anti lg 8.63		Jacobson et al. (2019)
9 ATL 313 (evodenoson)	Anti lg 9.15		Jacobson et al. (2019)
LASSBio-294	9,500		da Silva et al. (2017)
PSB-15826	14.8 human recombinant		De Filippo et al. (2016)
PSB-12404		IC50: 67	Fuentes et al. (2018)
PSB 16301		IC50: 5.5	Fuentes et al. (2018)
ATL-193	45.8 canine		Glover et al. (2001)
PSB-033	44		El-Tayeb et al. (2011)
CV 1808	190		Cunha et al. (1996)
AMP597	56		Clark et al. (2000)
UK-432094	4.8		Xu et al. (2011)
LUF5834	28		Beukers et al. (2004)

IC50: in functional assays in µM.