Table 2. Cytostatic (GI50 and TGI) and Cytotoxic (LC50) Parameters of Active Compounds.
compounds |
|||||
---|---|---|---|---|---|
18 (NSC 764190) | 21 (NSC 751486) | 23 (NSC 751478) | 25 (NSC 764189) | ||
log GI50 | median | –4.94 | –5.49 | –5.31 | –5.30 |
delta | 1.63 | 0.58 | 1.25 | 0.00 | |
range | 2.57 | 0.85 | 1.44 | 0.00 | |
log TGI | median | –4.00 | –5.10 | –5.12 | –5.30 |
delta | 0.22 | 0.22 | 0.00 | 0.00 | |
range | 0.22 | 0.62 | 0.00 | 0.00 | |
log LC50 | median | –4.00 | –4.80 | –5.12 | –5.30 |
delta | 0.00 | 0.18 | 0.00 | 0.00 | |
range | 0.00 | 0.28 | 0.00 | 0.00 |