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. 2021 Jan 28;12(2):288–294. doi: 10.1021/acsmedchemlett.0c00668

Table 2. “Reverse” Amide SAR.

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a

Data reported as average of ≥3 test results. See Supporting Information for description of assay conditions.

b

Data reported as average of ≥2 test results. See Supporting Information for description of assay conditions.

c

Percentage of the parent compound (0.5 μM) remaining after a 10 min incubation with 1 mg/mL of HLM or MsLM.