Table 2. “Reverse” Amide SAR.
Data reported as average of ≥3 test results. See Supporting Information for description of assay conditions.
Data reported as average of ≥2 test results. See Supporting Information for description of assay conditions.
Percentage of the parent compound (0.5 μM) remaining after a 10 min incubation with 1 mg/mL of HLM or MsLM.