. 2021 Feb 1;12(2):267–274. doi: 10.1021/acsmedchemlett.0c00647

Table 1. In Vitro Activity of 5–17 on FXR in a Hybrid Reporter Gene Assay^a.

Maximum relative activation corresponds to the activity of 1 μM GW4064 (1). Inactive indicates that there was no statistically significant reporter activation at the indicated concentration. Data are reported as mean ± SEM, n ≥ 3.

Table 1. In Vitro Activity of 5–17 on FXR in a Hybrid Reporter Gene Assaya.

Table 1. In Vitro Activity of 5–17 on FXR in a Hybrid Reporter Gene Assay^a.