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. Author manuscript; available in PMC: 2021 Feb 15.
Published in final edited form as: Pharmacol Ther. 2019 Feb 10;198:90–108. doi: 10.1016/j.pharmthera.2019.02.005

Table 1.

DPP4 intact substrates, and their amino acid sequences

Substrate Amino acid sequence Ref.
GLP-1(7–36) HA ↑ EGTFTSDVSSYLEGQAAKEFIAWLVKGR Orskov, Bersani, Johnsen, Hojrup, and Holst (1989))
GIP(1–42) YA ↑ EGTFISDYSIAMDKIHQQDFVNWLLAQKGKKNDWKHNITQ (Sparre-Ulrich et al. (2017))
PYY(1–36) YP ↑ IKPEAPGEDASPEELNRYYASLRHYLNLVTRQRY Grandt et al. (1994))
NPY(1–36) YP ↑ SKPDNPGEDAPAEDMARYYSALRHYINLITRQRY Tatemoto (1982)
CXCL12α(1–67) KP ↑ VSLSYRCPCRFFESHVARANVKHLKILNTPNCALQIVARLKNNNRQVCIDPKLKWIQEYLEKALNK Dong et al. (2012)

↑ DPP4 proteolytic site