Table 1.
DPP4 intact substrates, and their amino acid sequences
| Substrate | Amino acid sequence | Ref. |
|---|---|---|
| GLP-1(7–36) | HA ↑ EGTFTSDVSSYLEGQAAKEFIAWLVKGR | Orskov, Bersani, Johnsen, Hojrup, and Holst (1989)) |
| GIP(1–42) | YA ↑ EGTFISDYSIAMDKIHQQDFVNWLLAQKGKKNDWKHNITQ | (Sparre-Ulrich et al. (2017)) |
| PYY(1–36) | YP ↑ IKPEAPGEDASPEELNRYYASLRHYLNLVTRQRY | Grandt et al. (1994)) |
| NPY(1–36) | YP ↑ SKPDNPGEDAPAEDMARYYSALRHYINLITRQRY | Tatemoto (1982) |
| CXCL12α(1–67) | KP ↑ VSLSYRCPCRFFESHVARANVKHLKILNTPNCALQIVARLKNNNRQVCIDPKLKWIQEYLEKALNK | Dong et al. (2012) |
↑ DPP4 proteolytic site