Table 3A.
Clinical trials of CD40 agonist therapy
Drug | Feature | Phase | Disease | Outcome | PMID/Identifier |
---|---|---|---|---|---|
CP-870,893 | Human mAb | 1 | Solid tumors | Safe; Effective | 17327609 |
1 | Advanced solid tumor | Safe; Little efficiency | 20855968 | ||
1 | Advanced pancreatic ductal adenocarcinoma | Safe a; Effective | 23983255 21436454 |
||
1b | Malignant pleural mesothelioma | Safeb | 26386124 | ||
1 | Metastatic melanoma | Safe c; Effective | 30288340 | ||
Dacetuzumab | Humanized mAb | 1 | Refractory NHL | Safe; Effective | 19636010 |
1 | CLL | Safe; Little efficiency | 20038235 | ||
1 | Advanced MM | Safe; Little efficiency | 20133895 | ||
Relapsed DLBCL | Safe d; Effective | 22775314 | |||
2 | Relapsed DLBCL | Safe; Effective | 24919462 | ||
2b | Relapsed DLBCL | Safe e; Not effective | 25651427 | ||
ChiLob 7/4 | Chimeric mAb | 1 | CD40-expressing solid tumors and DLBCL | Safe; Little efficiency | 25589626 |
ADC-1013 | Human mAb | 1 | Advanced solid tumors | Safe | 30664811 |
Selicrelumab | Human mAb | 1 | Solid tumors | Unpublished | NCT02665416 |
1 | Refractory B-cell NHL | Ongoing | NCT03892525 | ||
APX005M | Humanized mAb | 1 | Solid tumors | Not reported | NCT02482168 |
1/2 | NSCLC& melanoma | Ongoing | NCT03123783 | ||
2 | Rectal adenocarcinoma | Ongoing | NCT04130854 | ||
2 | Soft tissue sarcoma | Ongoing | NCT03719430 | ||
2 | Melanoma | Ongoing |
NCT04337931 NCT02706353 |
||
1 | Pediatric central nervous system tumors | Ongoing | NCT03389802 | ||
SEA-CD40 | Humanized mAb | 1 | Carcinoma | Ongoing | NCT02376699 |
CDX-1140 | Human mAb | 1 | Carcinoma | Ongoing | NCT04364230 |
1 | Advanced malignancies | Ongoing | NCT03329950 | ||
2141-V11 | Fc-engineered human mAb | 1 | Solid tumor & cancer of skin | Ongoing | NCT04059588 |
NG-350A | Ad-human CD40 mAb | 1 | Metastatic cancer & epithelial Tumor | Ongoing | NCT03852511 |
BPX101 | Autologous DC transduced with Ad-human CD40 | 1 | Metastatic castration-resistant prostate cancer | Safe; Effective | 28608115 |
Abbreviations: Ad-human mAb, adenovirus carrying agonistic human CD40 mAb gene; Ad-human CD40, adenovirus carrying human CD40 gene; CLL, chronic lymphocytic leukemia; DLBCL, diffuse large B-cell lymphoma; Fc, constant fragment; mAb, monoclonal antibody; MM, multiple myeloma; NHL, non-Hodgkin lymphoma; NSCLC, non-small cell lung cancer.
in combination with gemcitabine;
in combination with cisplatin & pemetrexed;
in combination with tremelimumab;
in combination with rituximab & gemcitabine;
in combination with R-ICE (rituximab, ifosfamide, carboplatin and etoposide).