TABLE 12.
Pharmacokinetic parameters of bentysrepinine, M8 and M9 in a multiple doses study (Study 02).
| Analyte | Urine | Feces | ||
|---|---|---|---|---|
| Cumulative Ae (μmol/L) | Cumulative %Fe (%) | Cumulative Ae (μmol/L) | Cumulative %Fe (%) | |
| Bentysrepinine | 24.4 (7.9) | 3.0 (1.0) | 37.4 (32.7) | 4.6 (4.0) |
| M8 | 222.6 (44.6) | 27.2 (5.5) | 105.1 (50.5) | 12.9 (6.2) |
| M9 | 20.2 (7.4) | 2.1 (1.2) | — | — |
The data are expressed as mean (SD). Ae: amount of drug excreted in urine or feces, %Fe: % of drug excreted in urine or feces.