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. 2021 Jan 23;10(2):223. doi: 10.3390/cells10020223

Table 2.

Summary of phase II/III clinical trials investigating immunotherapy in BC with results from TIL analysis available.

Trial (Design) Setting, BC Subtype Treatment Arms TIL Variable (Cutoff a) Outcomes Results b
Keynote-086 [87]
(II) e
Advanced, TNBC Pembrolizumab (2 cohorts) Binary (median) ORR
DCR
Combined cohort: OR for ORR = 1.26 (1.03–1.55),
p = 0.01; OR for CDR 1.22 (1.02–1.46), p = 0.01
Impassion-130 [86] (III) Advanced, TNBC NabP–Atezo
NabP–Pbo
Binary (10%) PFS
OS
Predictive for Atezo benefit only in PD-L1+:
PD-L1+/strTILs low→ PFS: HR 0.74 (0.54–1.03), p = 0.07, OS: HR 0.65 (0.41–1.02) p = 0.06.
PD-L1+/strTILs high → PFS: HR 0.53 (0.38–0.74), p < 0.005; OS: HR 0.57 (0.35–0.92), p = 0.02.
PD-L1-/strTILs high → PFS: HR 0.99 (0.62–1.57), p = 0.97; OS: HR 1.53 (0.76–3.08), p = 0.24
Keynote-119 (III) [89] Advanced, TNBC Pembro
CT PFC c
Continuous,
Binary (5%)
BOR
DCR
PFS
OS
Positive association with clinical outcomes only in Pembro arm (p < 0.05)
TILs <5% → Pembro vs. CT: median OS 5.9 vs. 8.8 months, HR 1.50 (1.14–1.97)
TILs ≥5% → Pembro vs. CT: median OS 12.5 vs. 11.3 months, HR 0.75 (0.59–0.96)
Panacea [11]
(Ib-II)
Advanced, HER2+ Trastuzumab–Pembro Continuous OR
DCR
Positive association with ORR (p = 0.006) and DCR (p = 0.0006)
KATE-2
(II-R) [90,91]
Advanced, HER2+ TDM1–Atezo
TDM1–Pbo
Binary (5%) PFS
OS
Borderline positive association with OS in the atezolizumab arm
TILs < 5% → Atezo vs. Placebo: mPFS 5.5 (3.9-9.6) vs NE (4.0-NE), HR 0.62 (0.37-1.03). 1-year OS 84.2% vs. 100%, HR 1.43 (0.51–4.01)
TILs ≥ 5% → Atezo vs. Placebo: mPFS 8.5 (6.2-NE) vs 5.3 (4.0-9.5). 1-year OS 90.8% vs. 83.5%, HR 0.55 (0.26–1.12)
GeparNuevo [80]
(II R)
Neoadjuvant, TNBC Durva d→ Durva–NabP→ Durva–EC
Pbo→ Pbo–NabP→ Pbo–EC
Continuous
Categorical (10%, and 60%)
pCR strTILs (continuous): positive association with pCR, no predictive for Durva benefit
OR 1.23 (1.04–1.6), p = 0.019 in Durva arm; OR = 1.39 (1.12–1.74), p = 0.003 in Placebo arm.
intTILs: increase between baseline and end of the window phase associated with Durva benefit. OR 9.36 (1.26–69.65) p = 0.029
NeoTRIPaPDL1 [85]
(III)
Neoadjuvant, TNBC Cb–NabP–Atezo
Cb–NabP
Binary (40%) pCR Positive association with pCR, no predictive role
Atezo arm: strTILs ≥40% vs. <40% → pCR 71.43% vs. 28.07%, p = 0.001
CT arm: strTILs ≥40% vs. <40% → pCR 63.16% vs. 33.9%, p = 0.009
No interaction with treatment arm.
GIADA [92]
(II)
Neoadjuvant, Luminal-B e EC→ Nivo–ET Continuous pCR Positive association with pCR (p < 0.001)

a When applicable; b 95% confidence intervals reported in parentheses; c single agent chemotherapy per physician’s choice: capecitabine, eribulin, gemcitabine, vinorelbine; d in a proportion of patients, durvalumab was administered as induction treatment in the window phase. e luminal-B = hormone receptor-positive/HER2-negative, Ki67 ≥ 20% and/or grade 3. Abbreviations: BC, breast cancer; TN, triple-negative; str/int-TILs, stromal/intratumoral tumor-infiltrating lymphocytes; ORR, overall response rate; DCR, disease control rate; OR, odds ratio; CI, confidence interval; R, randomized; HR, hazard ratio; pCR, pathologic complete response, BOR, best overall response; (m)PFS, (median) progression-free survival; OS, overall survival; DCR, disease control rate; CT, chemotherapy; NabP, nab-paclitaxel; Pbo, placebo; Pembro, pembrolizumab; Atezo, atezolizumab; Cb, carboplatin; Durva, durvalumab; EC, epirubicin–cyclophosphamide; Nivo, nivolumab; ET, endocrine therapy.