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. 2021 Feb 10;22(4):1763. doi: 10.3390/ijms22041763

Table 2.

Selection of Free Fatty Acid Receptor 1 (FFAR1) allosteric ligands.

Name Structure References
Partial allosteric agonists
TAK-875/fasiglifam graphic file with name ijms-22-01763-i001.jpg Takeda Pharmaceuticals [70,71,78]
AM 837 graphic file with name ijms-22-01763-i002.jpg Amgen [62,79]
MK8666 graphic file with name ijms-22-01763-i003.jpg Merck [68,80,81,82]
Full allosteric agonists
AM 1638 graphic file with name ijms-22-01763-i004.jpg Amgen [62,83]
AP8 graphic file with name ijms-22-01763-i005.jpg Merck [81]
Compound 1 graphic file with name ijms-22-01763-i006.jpg Eli Lilly [84]