Table 3.
Antiproliferative activity of the lead compounds and paclitaxel against several human ovarian tumor cell lines.
Antiproliferative Activity IC50 (nM) | |||||
---|---|---|---|---|---|
Compound | SKOV3 | IGROV-1 | A2780 | OVCAR-8 | OVCAR-3 |
38 | 46 | 248 | 68 | 74 | 31 |
42 | 7 | 400 | 42 | 37 | 72 |
45 | 48 | 492 | 104 | 48 | 58 |
Paclitaxel 1 | 81 | 39 | 3 | 6 | 17 |
1 IC50 values against A2780, OVCAR-8, and OVCAR-3 cell lines from Bicaku, E. et al. evaluation [14].