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. Author manuscript; available in PMC: 2021 Mar 2.
Published in final edited form as: Annu Rev Immunol. 2020 Jan 21;38:341–363. doi: 10.1146/annurev-immunol-100819-121537

Table 1.

PHD inhibitors in preclinical models

PHI Model Year Reference
DMOG DSS colitis 2008 156
DSS colitis 2011 166
Radiation injury 2014 167
TNF-ΔARE ileitis 2010 158
Clostridium difficile infection 2010 59
Indomethacin-induced gastritis 2011 168
Pseudomonas aeruginosa infection 2013 169
Contact dermatitis 2019 142
Oral Fusobacterium infection 2019 170
Eosinophilic esophagitis 2019 23
Periodontitis 2018 171
FG-4497 TNBS colitis 2008 157
EtOH-induced liver disease 2019 172
AKB-4924 TNBS colitis 2014 159
TNF-ΔARE ileitis 2014 159
TRC160334 TNBS/DSS colitis 2014 173

Abbreviations: DMOG, dimethyloxalylglycine; DSS, dextran sodium sulfate; TNBS, trinitrobenzenesulfonic acid.