Table 4.
Data from direct FP binding experiments; N.D.: not determined; The results are presented as mean ± standard error.
Targeting WDR5 | EC50 (μM) | Ki (μM) |
---|---|---|
D206115-CRTLPFHEC | 5.9 ± 0.2 | 1.2 ± 0.04 |
D206116-CEKMVATHC | N.D. | N.D. |
D206179-CRTLPWNNC | 2.3 ± 0.6 | 0.5 ± 0.1 |
D206180-CRTLPYGAC | 2.7 ± 0.2 | 0.5 ± 0.05 |
D206181-CRTLPFGSC | 4.4 ± 0.4 | 0.9 ± 0.08 |