Table 2.
A few known kinase inhibitors
Drug candidate | Molecular target |
---|---|
Baricitinib | JAK1/2/3 |
BMS-986165 | Tyk2 |
Decernotinib | JAK-3 |
Delgocitinib | pan inhibitor of JAKs |
Fedratinib | JAK-2 |
Filgotinib | JAK-1 |
Itacitinib | JAK-1 |
NDI-031232 | Tyk2 |
NDI-031407 | Tyk2 |
Olacitinib | JAK1/2/3 |
Peficitinib | JAK-1/2/3 |
PF-06651600 | JAK-3 |
PF-06826647 | Tyk2/JAK-1/2 |
Ruxolitinib | JAK1/2 |
SAR-20347 | Tyk2/JAK-1/2/3 |
Solcitinib | JAK-1 |
Tofacitinib | JAK1/3 |
Upadacitinib | JAK-1 |