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. 2021 Mar 25;12:1875. doi: 10.1038/s41467-021-22084-5

Table 3.

Azidocarbonylation of indoles and their analogues to synthesize indole-3-carbonyl azidesa.

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aReaction conditions: KAP-Pd-PEPPSI-3 (5 mol%), indole (0.25 mmol), I2 (0.5 mmol), DABCO (0.5 mmol), CsF (1.0 mmol), DMF (2.0 mL), CO (2.0 MPa), 80 °C, 24 h. Then NaN3 (1.0 mmol) was added, room temperature, 7 h, isolated yield.

b30 h.

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