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. 2020 Feb 10;63(5):2588–2619. doi: 10.1021/acs.jmedchem.9b01526

Scheme 5. Synthesis of Compound 9d.

Scheme 5

Reagents and conditions: (a) HOBt (1.1 equiv), EDC (1.1 equiv), TEA (2.2. equiv) DCM, rt, 16 h, yield 42%.