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. 2021 Apr 8;21(9):548–569. doi: 10.1038/s41577-021-00524-z

Table 2.

Compound structures of described cGAS inhibitors

Compound Structure Ref.
PF-06928215 graphic file with name 41577_2021_524_Figb_HTML.gif 160
RU.365 graphic file with name 41577_2021_524_Figc_HTML.gif 12
RU.521 graphic file with name 41577_2021_524_Figd_HTML.gif 12
G150 graphic file with name 41577_2021_524_Fige_HTML.gif 161
Compound S3 graphic file with name 41577_2021_524_Figf_HTML.gif 163
Hydroxychloroquine graphic file with name 41577_2021_524_Figg_HTML.gif 164
Quinacrine graphic file with name 41577_2021_524_Figh_HTML.gif 164
X6 graphic file with name 41577_2021_524_Figi_HTML.gif 166
Suramin graphic file with name 41577_2021_524_Figj_HTML.gif 168
CU-76 graphic file with name 41577_2021_524_Figk_HTML.gif 162

cGAS, cyclic GMP–AMP synthase.