Table 3.

AlphaScreen counter assay.

Compound	Concentration (M)	% Binding
3478	5.00 × 10-5	98.39
	1.67 × 10-5	96.40
	5.56 × 10-6	97.72
	1.85 × 10-6	97.84
	6.17 × 10-7	103.76
	2.06 × 10-7	95.81
	6.86 × 10-8	102.51
	2.29 × 10-8	101.85
	7.62 × 10-9	102.56
	2.54 × 10-9	101.61
DMSOa	–	98.67

^aThe concentration of DMSO control was 1% v/v.