Table 10. X-ray Crystal Structures of Human MTHFDs.
| protein | ligands | resolution (Å) | PDB ID | refs |
|---|---|---|---|---|
| MTHFD1 | NADP | 1.50 | 1A4I | (211) |
| NADP, LY249543 | 2.20 | 1DIA | (212) | |
| NADP, LY345899 | 2.70 | 1DIB | ||
| NADP, LY374571 | 2.20 | 1DIG | ||
| NADP, LY249543 | 2.20 | 6ECP | (213) | |
| NADP, LY345899 | 2.70 | 6ECQ | ||
| NADP | 2.20 | 6ECR | ||
| MTHFD2 | NAD, LY345899 | 1.89 | 5TC4 | (209) |
| DS44960156 | 2.25 | 6JIB | (210) | |
| compound 1 | 2.50 | 6JID | ||
| DS18561882 | 2.25 | 6KG2 | (186) | |
| MTHFD1L | NA | NA | NA | NA |
| MTHFD2L | NA | NA | NA | NA |
NA, not applicable