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. 2021 Mar 1;4(2):624–646. doi: 10.1021/acsptsci.0c00223

Table 10. X-ray Crystal Structures of Human MTHFDs.

protein ligands resolution (Å) PDB ID refs
MTHFD1 NADP 1.50 1A4I (211)
  NADP, LY249543 2.20 1DIA (212)
  NADP, LY345899 2.70 1DIB
  NADP, LY374571 2.20 1DIG
  NADP, LY249543 2.20 6ECP (213)
  NADP, LY345899 2.70 6ECQ
  NADP 2.20 6ECR
         
MTHFD2 NAD, LY345899 1.89 5TC4 (209)
  DS44960156 2.25 6JIB (210)
  compound 1 2.50 6JID
  DS18561882 2.25 6KG2 (186)
         
MTHFD1L NA NA NA NA
         
MTHFD2L NA NA NA NA
a

NA, not applicable