Table 1.

List of X-ray crystallographic structures containing TAFI or activated TAFI (TAFIa) in the Protein Data Bank (PDB).

Form	PDB ID	TAFI Variant 1	Ligand 2	Resolution (A)	Ref.
TAFI	3D66	Human TAFI	-	3.1	[30]
	3D67	Human TAFI	GEMSA	3.4	[30]
	3D68	Human TAFI-IIYQ	-	2.8	[30]
	4P10	Human TAFI	Compound 5	2.0	[33]
	3DGV	Bovine TAFI	-	2.5	-
	3OSL	Bovine TAFI	TCI	6.0	[34]
	5HVF	Human TAFI-CIIYQ	Nanobody VHH-i83	2.8	[35]
	5HVG	Human TAFI-CIIYQ	Nanobody VHH-a204	3.0	[35]
	5HVH	Human TAFI-CIIYQ	VHH-i83 + VHH-a204	3.0	[35]
TAFIa	3D4U	Bovine TAFIa	TCI	2.5	[36]
	3LMS	Human TAFIa	TCI	1.7	[32]
	4UIA	Porcine TAFIa	Compound 3a	2.2	[37]
	4UIB	Porcine TAFIa	Compound 3p	1.9	[37]
	5LYF	Porcine TAFIa	Urea lead of compounds 1 and 6–7a	2.0	[38]
	5LYD	Porcine TAFIa	Compound 1	2.0	[38]
	5LYI	Porcine TAFIa	Compound 7a	1.6	[38]
	5LYL	Porcine TAFIa	Compound 6a	1.8	[38]

¹ TAFI-IIYQ: TAFI-T325I-T329I-H333Y-H335Q; TAFI-CIIYQ: TAFI-S305C-T325I-T329I-H333Y-H335Q. ² GEMSA: (2-guanidinoethylmercapto)-succinic acid; TCI: tick carboxypeptidase inhibitor.