. 2021 Mar 8;12(4):631–639. doi: 10.1021/acsmedchemlett.1c00029

Table 2. Chemical Structures of GW9662 Derivatives, Their RORγt Ligation, IC₅₀ ± SD (nM) (Data Recorded in Triplicate in Two Independent Experiments) And Full/Partial Inverse Agonistic Character^a.

Abbreviations: inv. ago., inverse agonist; rem. act., remaining activity; n.d., not determined.

Table 2. Chemical Structures of GW9662 Derivatives, Their RORγt Ligation, IC50 ± SD (nM) (Data Recorded in Triplicate in Two Independent Experiments) And Full/Partial Inverse Agonistic Charactera.