| ABC | ATP-binding cassette transporter |
| ADMA | asymmetric dimethylarginine |
| BCRP | breast cancer resistance protein |
| CrCl | creatinine clearance |
| CKD | chronic kidney disease |
| CMPF | 3-carboxy-4-methyl-5-propyl-2-furanopropanoic acid |
| CRF | chronic renal failure |
| DDI | drug–drug interaction |
| ENT1/SLC29A1 | equilibrative nucleoside transporter 1 |
| ENT2/SLC29A2 | equilibrative nucleoside transporter 2 |
| FDA | US Food and Drug Administration |
| GFR | glomerular filtration rate |
| GLUT9/SLC2A9 | facilitative glucose transporter 9 |
| GSA | guanidine succinate |
| GSH | glutathione |
| HNF1α/HNF1A | hepatocyte nuclear factor 1α |
| HNF4α/HNF4A | hepatocyte nuclear factor 4α |
| MATE1/SLC47A1 | multidrug and toxin extrusion protein 1 |
| MATE2/SLC47A2 | multidrug and toxin extrusion protein 2 |
| MATE2-K/SLC47A2 | multidrug and toxin extrusion protein 2 kidney-specific |
| MRP1/ABCC1 | multidrug resistance-associated protein 2 |
| MRP2/ABCC2 | multidrug resistance-associated protein 2 |
| MRP3/ABCC3 | multidrug resistance-associated protein 3 |
| MRP4/ABCC4 | multidrug resistance-associated protein 4 |
| MRP5/ABCC5 | multidrug resistance-associated protein 5 |
| MRP6/ABCC6 | multidrug resistance-associated protein 6 |
| MTX | methotrexate |
| NSAIDs | non-steroidal anti-inflammatory drugs |
| OAT1/SLC22A6 | organic anion transporter 1 |
| OAT2/SLC22A7 | organic anion transporter 2 |
| OAT3/SLC22A8 | organic anion transporter 3 |
| OAT4/SLC22A11 | organic anion transporter 4 |
| OATP1A2/SLCO1A2 | kidney organic anion transporting polypeptide 1A2 |
| OATP2B1/SLCO2B1 | kidney organic anion transporting polypeptide 2B1 |
| OATP4C1/SLCO4C1 | kidney organic anion transporting polypeptide 4C1 |
| OCT1/SLC22A1 | organic cation transporter 1 |
| OCT2/SLC22A2 | organic cation transporter 2 |
| OCT3/SLC22A3 | organic cation transporter 3 |
| OCTN1/SLC22A4 | organic cation/carnitine transporter 1 |
| OCTN2/SLC22A5 | organic cation/carnitine transporter 2 |
| OSTα/SLC51A | organic solute transporter α |
| OSTβ/SLC51B | organic solute transporter β |
| PAH | p-aminohippurate |
| PAN | puromycin aminonucleoside |
| PEPT1/SLC15A1 | peptide transporter 1 |
| PEPT2/SLC15A2 | peptide transporter 2 |
| P-gp. MDR1/ABCB1 | glycoprotein, multidrug resistance protein 1 |
| PMAT/SLC29A4 | plasma membrane amino-acid transporter |
| SGLT2/SLC5A2 | sodium-glucose co-transporter 2 |
| SLC | solute carrier |
| SLCO4A1/OATP4A1 | kidney organic anion transporting polypeptide 4A1 |
| URAT1/SLC22A12 | urate transporter 1 |
| XO | xanthine oxidase |