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. Author manuscript; available in PMC: 2021 Apr 30.
Published in final edited form as: J Med Chem. 2018 Oct 31;61(22):9908–9930. doi: 10.1021/acs.jmedchem.8b00639

Table 5.

Pharmacokinetic Parameters of 19a

mean ± SD
parameters iv (1 mg/kg)a ig (5 mg/kg)b
Tmax (h) 1.17 ± 0.76
Cmax (ng/mL) 23.5 ± 16
AUC0→t (h·ng/mL) 119 ± 10 89.7 ± 36
AUC0→∞ (h·ng/mL) 121 ± 10 109 ± 33
MRTINF (h) 1.01 ± 0.023 4.73 ± 3.3
T1/2 (h) 0.855 ± 0.011 3.08 ± 3.4
F (%) 15.5 ± 5.4
a

iv means intravenous injection.

b

ig means intragastrical administration.