Table 5.
Pharmacokinetic Parameters of 19a
mean ± SD |
||
---|---|---|
parameters | iv (1 mg/kg)a | ig (5 mg/kg)b |
Tmax (h) | 1.17 ± 0.76 | |
Cmax (ng/mL) | 23.5 ± 16 | |
AUC0→t (h·ng/mL) | 119 ± 10 | 89.7 ± 36 |
AUC0→∞ (h·ng/mL) | 121 ± 10 | 109 ± 33 |
MRTINF (h) | 1.01 ± 0.023 | 4.73 ± 3.3 |
T1/2 (h) | 0.855 ± 0.011 | 3.08 ± 3.4 |
F (%) | 15.5 ± 5.4 |
iv means intravenous injection.
ig means intragastrical administration.