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. Author manuscript; available in PMC: 2021 Apr 30.
Published in final edited form as: Curr Med Chem. 2013;20(28):3500–3514. doi: 10.2174/0929867311320280007

Table 2.

Targeted-NP-Based Therapeutics which Follow Active Targeting

Trade name NP Type Company Targeting Ligand Disease Payload Current
Status
Clinical Trial No.
SGT-53 Liposome SynerGene Therapeutics, Inc. Transferrin single-chain antibody fragment Advanced solid tumors Gene 53 Phase Ib NCT00470613
MBP-426 Liposome Mebiopharm Transferrin Solid tumors and esophagus disorders Oxaliplatin Phase II NCT00355888, NCT00964080
SEL-068 Polymeric Selecta Biosciences Small molecule Smoking cessation vaccine Nicotine antigen T-helper cell peptide, TLR agonist Phase I NCT01478893
CALAA-01 Polymeric Calando Human Transferrin Solid tumors siRNA Phase Ib NCT00689065
BIND-014 Polymeric Bind Biosciences PSMA peptide Metastatic cancer Docetaxel Phase I NCT01300533
SGT-94 Liposome SynerGene Therapeutics, Inc Anti-transferrin receptor single chain antibody fragment Solid tumors RB94 gene Phase I NCT01517464