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. 2021 Mar 25;23:e3. doi: 10.1017/erm.2021.5

Table 1.

Immunotherapeutic drugs approved by FDA (1997–2019)

Drug Description Mechanism First FDA approval
Atezolizumab Humanised Anti-PDL1 Checkpoint inhibition 2016
Avelumab Human anti-PDL1 Checkpoint inhibition 2017
Axicabtagene ciloleucel CAR-T cell anti-CD19 Neoantigen recognition 2017
Bevacizumab Humanised anti-VEGF Target therapy (anti-angiogenic effect) 2004
Blinatumomab Bispecific murine anti-CD19 and anti-CD3 Neoantigen recognition 2014
Brentuximab vedotin Chimeric anti-human CD30 (antibody-drug conjugate) Neoantigen recognition 2011
Cemiplimab Human anti-PD1 Checkpoint inhibition 2018
Cetuximab Chimeric anti-EGFR Target therapy (tumour anti-proliferative effect) 2004
Daratumumab Human anti-CD38 Neoantigen recognition
Immunomodulation
2015
Denosumab Humanised anti-RANKL Immunomodulation (anti-osteoclast activity) 2010
Dinutuximab Chimeric anti-GD2 Neoantigen recognition 2015
Durvalumab Human anti-PDL1 Checkpoint inhibition 2017
Elotuzumab Humanised anti-SLAMF7 Neoantigen recognition 2015
Gemtuzumab ozogamicin Humanised anti-CD33 (antibody-drug conjugate) Neoantigen recognition Target therapy 2001
Ibritumomab tiuxetan Murine anti-CD20 type II (radionuclide-linked Ab) Neoantigen recognition Target therapy 2002
Inotuzumab ozogamicin Humanised anti-CD22 (antibody-drug conjugate) Neoantigen recognition 2017
Ipilimumab Human anti-CTLA4 Checkpoint inhibition 2011
Necitumumab Human anti-EGFR Neoantigen recognition Target therapy (tumour anti-proliferative effect) 2015
Nivolumab Human anti-PD1 Checkpoint inhibition 2014
Obinutuzumab Humanised anti-CD20 type II Neoantigen recognition 2013
Ofatumumab Human anti-CD20 type I Neoantigen recognition 2010
Panitumumab Human anti-EGF Target therapy (tumour anti-proliferative effect) 2006
Peginterferon alfa-2b Immune modulator, anti-proliferative and anti-viral Immunomodulation 2011
Pembrolizumab Humanised anti-PD1 Checkpoint inhibition 2014
Pertuzumab Humanised anti-HER2 Neoantigen recognition 2012
Polatuzumab vedotin Humanised anti-CD79b (Ab-drug conjugate) Neoantigen recognition Target therapy 2019
Ramucirumab Human anti-VEGFR-2 Target therapy (anti-angiogenic effect) 2014
Rituximab Chimeric anti-CD20 type I Neoantigen recognition 1997
Sipuleucel-t PAP-specific APC based vaccine Neoantigen recognition 2010
Tisagenlecleucel CAR-T cell anti-CD19 Neoantigen recognition 2017
Tositumomab Radionuclide-linked murine anti-CD20 type II Neoantigen recognition Target therapy 2003
Trastuzumab Humanised anti-HER2 Neoantigen recognition 1998
Trastuzumab emtansine Humanized anti-HER2 (conjugated antibody) Neoantigen recognition 2013
Tremelimumab Human anti-CTLA4 Checkpoint inhibition 2015

Record of immunotherapeutic drugs approved by the FDA (www.fda.gov) for the treatment of several cancer types and their mechanism of action (data updated until 31/Dec/2019).