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. Author manuscript; available in PMC: 2021 Jul 23.
Published in final edited form as: J Med Chem. 2020 Jul 7;63(14):7695–7720. doi: 10.1021/acs.jmedchem.0c00520

Table 7.

Inhibition of CH-σ Interactions by Representative Compounds

no. MIC μg/mL) IC50 (μM) no. MIC (μg/mL) IC50 (μM)
33   16 67.0 ± 4.7 44 8 42.9 ± 2.5
37 256 97.0 ± 9.6 45 4 15.0 ± 0.7
43     4 11.6 ± 0.6 55 8 25.1 ± 1.5