Table 1.
Average Percent Protonation of Lumefantrine in ASDs (n = 3).
| Sample | % Protonation |
|---|---|
| 2:8 Lum:HPMCP | 42 ± 3 |
| 3:7 Lum:HPMCP | 40 ± 2 |
| 4:6 Lum:HPMCP | 37 ± 3 |
| 2:8 Lum:HPMCAS | 37 ± 4 |
| 3:7 Lum:HPMCAS | 35 ± 7 |
| 4:6 Lum:HPMCAS | 14 ± 2 |
| 4:6 Lum:CAP | 32 ± 2 |
| 4:6 Lum:EL100 | 38 ± 4 |
| Amorphous lumefantrine | 3 ± 1 |