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. 2021 Jun;110(6):2423–2431. doi: 10.1016/j.xphs.2020.12.033

Table 1.

Average Percent Protonation of Lumefantrine in ASDs (n = 3).

Sample % Protonation
2:8 Lum:HPMCP 42 ± 3
3:7 Lum:HPMCP 40 ± 2
4:6 Lum:HPMCP 37 ± 3
2:8 Lum:HPMCAS 37 ± 4
3:7 Lum:HPMCAS 35 ± 7
4:6 Lum:HPMCAS 14 ± 2
4:6 Lum:CAP 32 ± 2
4:6 Lum:EL100 38 ± 4
Amorphous lumefantrine 3 ± 1