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. 2021 Mar 12;11(5):1158–1174. doi: 10.1016/j.apsb.2021.03.013

Table 2.

Delivery strategies for different types of agents.

Category of agents Agent Formulation Ref.
Small molecule Dexamethasone PEG‒Dex conjugates 19
Methotrexate Dextran sulfate‒MTX conjugates 20
Methotrexate Albumin‒MTX conjugates 21
Methylprednisolone Cyclodextrin‒α-methylprednisolone conjugates 22
Dexamethasone PEGylation liposomes 23
Dexamethasone DC8,9PC and DSPE-PEG liposomes 24
Dexamethasone PCL‒PEG micelles 25
Methotrexate SA-Dex-OA/MTX micelles 26
Curcumin HA-Cur micelles 27
Methotrexate MTX-loaded albumin nanoparticles 28
Methotrexate Au/Fe half-shell PLGA nanoparticles 29
Nucleic acid IL-1β siRNA Lipidoid‒polymer hybrid nanoparticles 30
p65 siRNA PCL‒PEI and PCL‒PEG micelles 31
siRNA against BTK PEG-b-PLGA nanoparticles 32
TNF-α siRNA PEGylated solid-lipid nanoparticles 33
Peptide/protein Core peptide PEGylated liposomes 34
TNF-α antibody Carboxymethyl cellulose microneedle 35
Etanercept HA crosslinked microneedle 36
TRAIL HSA‒TRAIL conjugates 37
Tocilizumab Gold nanoparticles 38

PEG, polyethylene glycol; DC8,9PC, 1,2-bis (10,12-tricosadiynoyl)-sn-glycero-3-phosphocholine; PCL‒PEG, poly(ethylene glycol)‒poly(ε-caprolactone); SA, sialic acid; OA, octadecanoic acid; PCL‒PEI, poly(ε-caprolactone)-polyetherimide; HA, hyaluronic acid; Cur, curcumin; PLGA, poly(lactic-co-glycolic acid); TRAIL, tumor necrosis factor (TNF)-related apoptosis-inducing ligand; HSA, human serum albumin.