Table 3.
R2 | R1 | k1 (h−1) | k2 (h−1) | tcompl | Yield (%) |
---|---|---|---|---|---|
Me | H | 2.67 | 0.70 | 5.5 h | 95 |
Et | H | 0.88 | 0.27 | 9.5 h | 90 |
iPr | H | 2.08 | 1.33 | 4.5 h | 99 |
Bn | H | 23.8 | 9.36 | 45 min | 80 |
Et | Me | 0.86 | 0.16 | 17.5 h | 87 |
Et | MeC(O) | 0.90 | 0.35 | 8.5 h | 86 |
R2 | R1 | k1 (h−1) | k2 (h−1) | tcompl | Yield (%) |
---|---|---|---|---|---|
Me | H | 2.67 | 0.70 | 5.5 h | 95 |
Et | H | 0.88 | 0.27 | 9.5 h | 90 |
iPr | H | 2.08 | 1.33 | 4.5 h | 99 |
Bn | H | 23.8 | 9.36 | 45 min | 80 |
Et | Me | 0.86 | 0.16 | 17.5 h | 87 |
Et | MeC(O) | 0.90 | 0.35 | 8.5 h | 86 |