Construction of diverse peptide structural architectures via chemoselective peptide ligation

. 2021 Apr 13;12(20):7091–7097. doi: 10.1039/d1sc01174j

Entry	Sequence	%
12	H-SDKITED′A-NH₂	>98^b, 42.3^c
13	H-SNKQARD′KIYQSQT-NH₂	95.2^b, 46.1^c

D′ = Asp(benzofuran), (K–S) = Lys–Ser dipeptide, SAL = salicylaldehyde.

Percentage conversion to product based on UPLC-MS analysis of the crude reaction mixture.

Isolated yield based on ligation.