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. 2021 Apr 23;6(17):11375–11388. doi: 10.1021/acsomega.1c00360

Table 4. Percentage of PANC-1Cell Survival Studies with SAHA Derivatives.

  concentrations
 
entry 3.125 μM 6.25 μM 12.5 μM 25.0 μM 50.0 μM IC50 (μg/mL)
4a 90.76 ± 0.95 83.52 ± 0.54 75.77 ± 1.06 63.93 ± 0.87 58.42 ± 0.72 57.08
4b 92.61 ± 0.46 84.88 ± 0.59 76.86 ± 0.73 64.87 ± 0.63 57.67 ± 0.78 55.66
4c 93.78 ± 1.27 85.69 ± 0.19 74.36 ± 0.49 67.58 ± 0.23 63.92 ± 0.57 67.21
4d 94.42 ± 0.78 88.69 ± 0.65 81.93 ± 0.52 76.58 ± 0.37 72.66 ± 0.48 218.16
4e 99.91 ± 0.85 96.33 ± 0.56 94.25 ± 0.79 92.18 ± 0.83 89.71 ± 0.65 258.74
4f 99.41 ± 0.38 97.75 ± 0.54 96.13 ± 0.42 94.76 ± 0.37 91.85 ± 0.59 332.59
4g 98.02 ± 0.55 91.15 ± 0.73 89.60 ± 0.41 88.04 ± 0.39 85.50 ± 0.65 221.08
4h 95.71 ± 0.48 91.58 ± 0.43 89.13 ± 0.37 88.01 ± 0.62 86.05 ± 0.53 262.37
4i 99.54 ± 0.75 95.69 ± 0.66 90.47 ± 0.62 88.89 ± 0.59 85.97 ± 0.79 188.16
4j 97.33 ± 0.98 93.67 ± 0.87 89.43 ± 0.76 84.69 ± 0.65 79.54 ± 0.93 129.54
4k 88.15 ± 0.65 82.26 ± 0.48 74.86 ± 0.35 66.52 ± 0.39 54.92 ± 0.52 54.31
4l 99.87 ± 0.63 93.14 ± 0.87 87.28 ± 0.74 82.27 ± 0.35 77.54 ± 0.72 110.24