Skip to main content
. 2021 Apr 10;64(8):4312–4332. doi: 10.1021/acs.jmedchem.0c01002

Table 3. Selectivity Data for Bicyclic n-Carboxylic Acids.

  hGPR120
hGPR40
comp. EC50a (Ca2+) EC50 (β-arr) EC50 (IP1) EC50 (Ca2+) EC50 (β-arr) EC50 (IP1)
23 -b - 63 - - 1828
24 - 24 35 - - >10000
25 - 84 220 - - >10000
26 - 66 98 - - >10000
27 93 - - >100000 - -
28 740 - - >100000 - -
29 360 - - >100000 - -
a

nM.

b

Data not registered for the referred compound.