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. 2021 Apr 10;64(8):4312–4332. doi: 10.1021/acs.jmedchem.0c01002

Table 4. Selectivity Data for Nonacidic Head Derived Compounds.

  hGPR120
 hGPR40
comp. EC50a/pEC50d (Ca2+) EC50/pEC50d (β-arr) EC50/pEC50d (Ca2+) EC50/pEC50d (β-arr)
30 165 125 -c -
31 6.3d - <4.5d -
32 6.63d 6.91d NAb -
33 120 5.2 - -
a

nM.

b

NA: not active at 100 μM.

c

Data not registered for the referred compound.

d

pEC50 value.