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. 2021 Mar 25;64(7):3508–3545. doi: 10.1021/acs.jmedchem.0c01808

Table 4. Activity in Vitro of 56 against Laboratory Strains of HIV-1a.

2.6.

coreceptor tropism virus EC50 [nM]
CCR5 JR-FL 0.4 ± 0.1
  SF-162 0.5 ± 0.2
  Bal 1.7 ± 0.5
CXCR4 LAI 0.7 ± 0.4
  NL4-3 2.2 ± 0.6
  MN 14.8 ± 5.2
  IIIb 16.2 ± 1.7
  RF >2000
a

Data are taken from Meanwell et al.15