. 2021 Mar 25;64(7):3508–3545. doi: 10.1021/acs.jmedchem.0c01808

Table 5. GIIA and GIB PLA₂ Inhibition by Indole-3-glyoxamides 59–62^a.

cpd	R₁	R₂	hGIIA PLA₂ [μM]	hGIB PLA₂ [μM]	pGIB PLA₂ [μM]
59	2-(C₆H₅)C₆H₄CH₂	CH₃	0.006 ± 0.001	0.364	0.097
60	3-(C₆H₅)C₆H₄CH₂	CH₃	0.009 ± 0.001	0.57	0.007
61	C₆H₅CH₂	CH₃	0.011 ± 0.004	0.761	0.015
62			0.009 ± 0.001	0.228	0.048

Data are taken from Draheim et al.¹²²

Table 5. GIIA and GIB PLA2 Inhibition by Indole-3-glyoxamides 59–62a.