Table 6. GIIA Inhibition by Indolizine-3-glyoxamide Derivativesa.
| cpd | hGIIA PLA2 [μM] chromogenic assay | hGIIA PLA2 [μM] PC/DOC assay |
|---|---|---|
| 63 | 0.006 | 0.003 |
| 64 | 0.008 | 0.0014 |
| 65 | 0.007 | 0.007 |
| 66 | 1.1 | b |
| 67 | 19 | b |
| 68 | >50 | b |
| 69 | 0.03 | 0.005 |
Data are taken from Hagishita et al.134
Value was not calculated for this compound.
