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. 2021 Mar 25;64(7):3508–3545. doi: 10.1021/acs.jmedchem.0c01808

Table 6. GIIA Inhibition by Indolizine-3-glyoxamide Derivativesa.

2.7.

cpd hGIIA PLA2 [μM] chromogenic assay hGIIA PLA2 [μM] PC/DOC assay
63 0.006 0.003
64 0.008 0.0014
65 0.007 0.007
66 1.1 b
67 19 b
68 >50 b
69 0.03 0.005
a

Data are taken from Hagishita et al.134

b

Value was not calculated for this compound.