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. 2021 Mar 25;64(7):3508–3545. doi: 10.1021/acs.jmedchem.0c01808

Table 8. Inhibitory Activity of Peptidyl Derivatives against Norovirus 3CLpro in Vitro (IC50) and in Cell-Based Replicon System (ED50)a.

3.2.1.

cpd IC50 [μM] ED50 [μM]
97 1.45 7.8
98 2.1 0.8
99 2.3 0.9
a

Data taken from Mandadapu et al.187