Table 4. Kinase Selectivity of Compound 27.
| kinase | IC50 (μM) |
|---|---|
| BTK | 0.142 |
| BMX | 0.129 |
| LCK | 0.130 |
| ErbB4 | 0.377 |
| TEC | 0.409 |
| TXK | 1.77 |
| FGR | 4.76 |
| B-RAF | 7.84 |
| SRC | 3.49 |
| HCK | >30 |
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