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. 2021 Apr 8;12(5):836–845. doi: 10.1021/acsmedchemlett.1c00113

Table 5. Pharmacokinetic Profiles of C5 in Rats.

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parameter p.o. (10 mg/kg) i.v. (2 mg/kg)
Kel (h–1) 0.232 ± 0.031 0.981 ± 0.263
Tmax (h) 2.17 ± 3.3  
T1/2 (h) 3.02 ± 0.38 0.74 ± 0.193
Cmax (ng/mL) 4499 ± 1754  
AUC0–t (ng/mL·h) 20 742 ± 4166 4601 ± 1684
AUC0–∞ (ng/mL·h) 26 943 ± 2245 4617 ± 1688
MRT (h) 5.58 ± 1.36 0.73 ± 0.21
F (%) 90.2 ± 18.1