Overall biodistribution results of 64Cu-Labeled HYR-4 and HYR-17 for the three time points evaluated (2, 60, and 240 min; % injected dose/gram, mean ± SEM).
Organ | HYR-4 | HYR-17 | ||||
---|---|---|---|---|---|---|
2 min | 60 min | 240 min | 2 min | 60 min | 240 min | |
Blood | 2.85 ± 0.52 | 1.02 ± 0.12 | 0.86 ± 0.10 | 26.82 ± 1.59 | 3.70 ± 0.06 | 1.24 ± 0.08 |
Lung | 3.77 ± 0.88 | 3.36 ± 0.25 | 4.47 ± 0.49 | 11.02 ± 0.52 | 3.65 ± 0.16 | 4.47 ± 0.49 |
Liver | 32.48 ± 3.94 | 8.84 ± 0.98 | 9.57 ± 1.19 | 11.50 ± 0.69 | 14.79 ± 1.71 | 12.16 ± 1.28 |
Kidney | 30.27 ± 0.44 | 9.39 ± 2.02 | 8.24 ± 1.95 | 15.96 ± 0.81 | 34.17 ± 2.87 | 21.40 ± 2.27 |
Muscle | 0.37 ± 0.08 | 0.30 ± 0.02 | 0.30 ± 0.04 | 0.89 ± 0.04 | 0.62 ± 0.02 | 0.45 ± 0.01 |
Brain | 0.16 ± 0.02 | 0.10 ± 0.01 | 0.15 ± 0.03 | 0.99 ± 0.04 | 0.20 ± 0.00 | 0.15 ± 0.02 |
Bone | 0.54 ± 0.11 | 0.45 ± 0.01 | 0.59 ± 0.07 | 1.59 ± 0.07 | 0.59 ± 0.09 | 0.64 ± 0.07 |
Tail | 15.91 ± 2.84 | 12.8 ± 5.38 | 3.69 ± 1.92 | 2.53 ± 0.16 | 3.20 ± 0.29 | 1.05 ± 0.05 |