Table 2. In Vitro Off-Target Profile of Lead Compound Z-Pst–l-Glu–Hph–NH2.
May1 C. neoformans | HIV-1 Pr wild-type | Pepsin porcine | Renin human | Cathepsin D human | Cathepsin E human |
---|---|---|---|---|---|
Ki 12 ± 1 nM | 32 ± 5 pM56 | 1.6 ± 0.3 μM | 19 ± 2 μM | 620 ± 50 nM | 440 ± 70 nM |