Table 1.
Inhibition data of CA isoforms I, II, IX, and XII by inhibitors ACTZ, AN6-277, and AN11-740 by a stopped flow CO2 hydrase assay29.
Cmpd | KI (nM)a |
|||
---|---|---|---|---|
CA I | CA II | CA IX | CA XII | |
ACTZ | 250 ± 15 | 12 ± 0.8 | 25 ± 1.4 | 5.7 ± 0.5 |
AN6-277b | 565.6 ± 34.2 | 1.2 ± 0.1 | 2.6 ± 0.2 | 1.1 ± 0.1 |
AN11-740 | 1580 ± 110c | 5.9 ± 0.4 c | 1.3 ± 0.1 | 3.0 ± 0.2 |