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. 2021 May 21;13(11):2541. doi: 10.3390/cancers13112541

Table 1.

TKIs KRAS G12C Inhibitors in Clinical Development.

Drug Sponsor Stage ClinicalTrials.gov Identifier
Sotorasib Amgen Phase I–III NCT04185883
Adagrasib Mirati Phase I–III NCT03785249
GDC-6036 Genentech/Roche Phase I NCT04449874
JNJ-74699157 Janssen Phase I NCT04006301
D-1553 Inventis Bio Phase I NCT04585035