Table 1.
TKIs KRAS G12C Inhibitors in Clinical Development.
| Drug | Sponsor | Stage | ClinicalTrials.gov Identifier |
|---|---|---|---|
| Sotorasib | Amgen | Phase I–III | NCT04185883 |
| Adagrasib | Mirati | Phase I–III | NCT03785249 |
| GDC-6036 | Genentech/Roche | Phase I | NCT04449874 |
| JNJ-74699157 | Janssen | Phase I | NCT04006301 |
| D-1553 | Inventis Bio | Phase I | NCT04585035 |