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. 2021 May 31;26(11):3309. doi: 10.3390/molecules26113309
Mycobacterium tuberculosis Mtb
H. proteasome Human proteasome
MIC Minimum inhibitory concentration
ACT Artemisinin-based combination therapies
aaRSAmino Acyl tRNA synthetase
CQ Chloroquine
ADME Absorption, distribution, metabolism, and excretion
SsrA-tagged protein Caseinolytic-protease-specific degradation protein
RLU Relative luminescence
WT cell lines Wild-type cell lines
aaRS Aminoacyl-tRNA synthetase
ClpP Caseinolytic proteases
TB Tuberculosis
Chloromethyl ketones CMKs
enoyl- reductase ENR
Enoyl-[acyl-carrier-protein] reductase [NADH] InhA
Nicotinamide adenine dinucleotide oxidized NAD+
Nicotinamide adenine dinucleotide reduced NADH
artemisinin-based combination therapies ACT
Plasmodium Falciparum P. Falciparum
Plasmodium falciparum 3D7 CQ-sensitive 3D7
structure−activity relationship studies SARs
3D7 Chloroquine (CQ) sensitive P. falciparum strain
W2 Chloroquine (CQ) resistant P. falciparum strain
D2d Chloroquine (CQ) resistant P. falciparum strain
half-life t1/2
availability F
WT cells Wild-type cells