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. 2021 May 7;12(6):991–995. doi: 10.1021/acsmedchemlett.1c00135

Table 4. Drug Concentrations in Fecal Samples of Selected Compounds.

  MIC, μg·mL–1a selectivityb dose, mg·kg–1 μg g–1 feces conc. feces/MIC
4 0.25 1 20 2.8 11
5c 0.125 128 20 13 108
87 0.125 1024 10 0.79 6.6
107 1 ≥256 20 2.4 2.4
108 1 64 20 49 49
116 0.50 128 20 3.7 7.4
a

C. difficile strain, ATCC 43255, ribotype 087.

b

Selectivity is defined as MICMRSA/MICC. difficile.

c

Reported previously; included for ease of comparison.