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. 2021 May 19;12(6):961–968. doi: 10.1021/acsmedchemlett.1c00233

Table 2. List of Receptors and Transporters Examined in the Dezocine Receptor Screening Panela.

serotonin receptors adrenoreceptors dopamine receptors
5-HT1A 5-HT2C α1A α2C D1
5-HT1B 5-HT3 α1B β1 D2
5-HT1D 5-HT5A α1D β2 D3
5-HT1E 5-HT6 α2A β3 D4
5-HT2A 5-HT7 α2B   D5
5-HT2B        
GABA receptors sigma receptors muscarinic receptors
GABA-A sigma 1 M1
rat benzodiazepine site sigma 2 M2
    M3
    M4
    M5
histamine receptors opioid receptors biogenic amine transporters
H1 μ-receptor serotonin
H2 κ-receptor norepinephrine
H3 δ-receptor dopamine
a

Taken from Liu et al., 2014.50