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. 2021 Jun 7;13(6):843. doi: 10.3390/pharmaceutics13060843

Table 4.

Applications of genetically modified MSCs in vivo.

Delivery System Carrier Nucleic Acid Cell Vehicles Application Model/Host Ref
Type Composition Vector Delivered Gene/siRNA
Non-viral Liposomes Lipofectamine Plus® Plasmid DNA hTERT MSC line derived from fetal porcine pancreas Hyperglycemia Diabetic model/Kunbai strain mice [113]
Polymer PEI Plasmid DNA TRAIL BM-MSCs Melanoma Melanoma model/e C57BL/6 mice [115]
Polymer Chitosan Plasmid DNA BMP-2 BM-MSCs Bone regeneration Calvarial defect model/Rats [85]
Polymer PEI Plasmid DNA BMP-2 BM-MSCs deriver MVs within gene-activated scaffold (DBM/MVs-PEI/phBMP2) Bone regeneration Femoral condylar defect/New Zealand white rabbits [86]
Polymer Alginate GAM Plasmid DNA BMP-2 Rat BM-MSCs Bone regeneration Orthotopic spinous process defect/Fischer 344 inbred rats [87]
Polymer LPEI Plasmid DNA VEGF BM-MSCs Myocardial infarction MI model/SD rats [95]
Polymer Cationized pullulan Plasmid DNA Suicide gene (CMV-TK) Rat BM-MSCs Melanoma Pulmonary melanoma metastasis model/C57BL6 mice [83]
Polymer LPEI Plasmid DNA CDY::UPRT AT-MSCs GDEPT: Chemo-resistant glioblastoma Temozolomide resistant U-251MG cells/Nude mice [116]
Polymers PEI-PLGA Plasmid DNA and siRNA coSOX9-pDNA/Cbfa-1-siRNA hMSCs encapsulated in fibrin hydrogels Chondrogenic differentiation Nude BALB/c mice [117]
Polymers PLL-PEI Plasmid DNA HSV-TK and TRAIL rMSCs Glioblastoma Glioma model/SD rats [101]
Polymeric NPs BA-PEI Plasmid DNA VEGF BM-MSCs Myocardial infarction MI model/SD rats [96]
Plasmid-activated scaffolds Chitosan-gelatin andnHA Plasmid DNA TGF-β1 and BMP-2 BM-MSCs Regeneration of articular cartilage and subchondral bone Knee ostochondral defect model/Rabbits [118]
nHA dual gene-activated scaffold nHA and PEI Plasmid DNA BMP-2 and VEGF rMSCs Bone regeneration Critical-sized cranial bone defect model/Rats [88]
Peptide conjugated NPs Cationic AuNPs and PEP Plasmid DNA VEGF Rat BM-MSCs Antimicrobial and wound healing properties Infected full thickness skin defect model/Mice [114]
Viral AAV IL-10 hBM-MSCs Cerebral ischemia MCAO I/R model/SD rats [82]
Adenovirus HSV-TK/GCV BM-MSCs Intracranial gliomas Intracranial human U87 glioma model/Nude mice [100]
Adenovirus HGF hBM-MSCs Spinal cord injury Spinal cord injury model/ SD rats [80]
Adenovirus EGFR Murine BM-MSCs Brain tumors Intracranial GL261 glioma or B16 melanoma/C57BL/6 mice [119]
Adenovirus IFN-β hBM-MSCs Pancreatic cancer Transplant PANC-1 cancer model/SCID mice [103]
Fiber-modified adenovirus kringle1-5/EGFP hPMSCs in Matrigel plugs Suppression of angiogenesis Subcutaneous cell loaded matrigel plugs/ BALB/c nude [105]
Gamma -Retrovirus IL7-IL12 hBM-MSCs Colorectal cancer Transplant LS174T colorectal cancer model/NSG mice [102]
Gamma-retrovirus HSV-TK hBM-MSCs Gastrointestinal/ hepatopancreatobiliary adenocarcinoma Phase I and II clinical trial [84]
HSV-1 HGF rBM-MSCs Cerebral ischemia MCAO I/R model/Wistar rats [81]
Lentivirus miR-126 BM-MSCs Myocardial infarction MI model/Mice [99]
Lentivirus HGF UCB-MSCs Myocardial infarction MI model/SCID mice [97]
Lentivirus FGF21 Mouse BM-MSCs Brain Injury Impact-induced traumatic brain Injury model/C57BL/6 mice [92]
Lentivirus CXCR4 rBM-MSCs Cerebral ischemia MCAO I/R model/SD rats [94]
Recombinant adenovirus VEGF BM-MSCs Cerebral ischemia MCAO I/R model/rats [93]
Retrovirus AKT Mouse BM-MSCs Myocardial infarction MI model/C57BL/6 mice [98]
Hybrid Adenovirus/liposome Ad-hEndo hPMSCs Ovarian cancer Transplant A2780 ovarian cancer model/ Nude mice [104]
Adenovirus/CPP stTRAIL hUCB-MSCs Glioblastoma Intracranial xenograft human glioma model/Athymic nude mice [120]
Adenovirus/4HP4 IL-12M rBM-MSCs Melanoma and cervical cancer B16F10 melanoma and TC-1 cervical cancer models/SCID mice [121]

Note: 4HP4: tetrameric form of cell-permeable peptide; CPP: cell-permeable peptide; HSV: herpes simplex virus; tTATop-BMP-2: tetracycline transactivator and BMP-2 cDNAs; BA-PEI: bile acid-modified polyethyleneimine; PMAA: polymethacrylate acid; CMV: cytomegalovirus; AT-MSCs: adipose tissue-derived MSCs; HIF-1 α: hypoxia-inducible factor-1α; CDY::UPRT: cytosine deaminase and uracil phosphoribosyl transferase; GAM: gene-activated matrix; GDEPT: gene-directed enzyme prodrug therapy; MVs: microvesicles; DBM: demineralized bone matrix; PLL-PEI: polylysine-modified polyethylenimine; hPMSCs: human placenta-derived MSCs; HSV: herpes simplex virus; MCAO I/R: middle cerebral artery occlusion ischemia/reperfusion; SD: Sprague-Dawley; MI: myocardial infarction; hEndo: human endostatin; UCB-MSCs: umbilical cord blood-derived MSCs.