Table 3.
Antiproliferative activity of target compounds against GBM cell lines (IC50, μM)a.
| COM. | U87 | U251 | T98G | U87-EGFRvIII |
|---|---|---|---|---|
| 1d | 63.28 ± 10.45 | 33.28 ± 3.36 | 20.62 ± 0.30 | 67.19 ± 3.20 |
| 1e | 53.61 ± 2.51 | 36.1 ± 2.53 | 20.07 ± 0.67 | >100 |
| 1q | 47.04 ± 3.78 | 30.02 ± 0.93 | 20.73 ± 0.67 | 68.98 ± 8.39 |
| 1s | 30.30 ± 0.84 | 24.61 ± 2.28 | 16.39 ± 2.12 | 50.46 ± 0.97 |
| PP2 | 39.94 ± 6.91 | 21.14 ± 2.16 | 12.52 ± 2.37 | 49.11 ± 7.76 |
aIC50 values are presented as mean values of at least three independent experiments.