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. 2021 Jun 2;64(12):7926–7962. doi: 10.1021/acs.jmedchem.0c02265

Table 1. IC50 Values of Compounds 16 on a Selected Panel of Cancer Cell Lines.

  IC50 (μM)a
Compd. NCI-H460 H1299 SKOV-3 DU145 MCF7 MCF10A MB-MDA-231 SF268 HT-29 HCT-15
1 40.52 >100 27.85 32.67 22.36 >100 57.12 >100 >100 >100
2 >100 >100 56.18 >100 >100 >100 >100 >100 >100 >100
3 >100 >100 >100 >100 >100 >100 >100 >100 >100 >100
4 44.77 >100 20.15 >100 41.34 >100 68.12 >100 >100 >100
5 >100 >100 >100 >100 88.1 >100 >100 >100 >100 >100
6 40.32 90.81 >100 13.06 16.75 88.63 21.60 38.8 36.42 54.12
a

Data from ref (101).